|
Benzopyranopyridine derivatives. 1. Aminoalkyl derivatives of the azaxanthenes as bronchodilating agents Frank J. Villani, Thomas A. Mann, Elizabeth A. Wefer, Janet Hannon, Louis L. Larca, Mildred J. Landon, William Spivak, Dhiru Vashi, Salvatore Tozzi, and et al. pp 1 - 8; DOI: 10.1021/jm00235a001 |
|
Carbocyclic prostaglandin analogs. 1. Steroid carboxylic acids D. L. Venton, R. E. Counsell, J. H. Sanner, and K. Sierra pp 9 - 16; DOI: 10.1021/jm00235a002 |
|
Aromatic amino acid hydroxylase inhibitors. 4. 3-Substituted .alpha.-methyltyrosines Ahmed H. El Masry, Souheir E. El Masry, Larry E. Hare, and Raymond E. Counsell pp 16 - 20; DOI: 10.1021/jm00235a003 |
|
Effect of acylation with eleostearic acids on the monoamine oxidase inhibitory potency of some hydrazine antidepressants in mice Song Y. Hsu, Chian L. Huang, and Irving W. Waters pp 20 - 23; DOI: 10.1021/jm00235a004 |
|
Comparison of the effects of histamine and tolazoline on adenylate cyclase activity from guinea pig heart Ira Weinryb and Inge M. Michel pp 23 - 26; DOI: 10.1021/jm00235a005 |
|
Synthesis and microbiological activities of some monohalogenated analogs of tyrosine Tommy J. McCord, David R. Smith, Douglas W. Winters, John F. Grimes, Karen L. Hulme, Lawrence Q. Robinson, Larry D. Gage, and Alvie L. Davis pp 26 - 29; DOI: 10.1021/jm00235a006 |
|
Charge-transfer constant. New substituent constant for structure-activity relations Bogumil Hetnarski and R. D. O'Brien pp 29 - 33; DOI: 10.1021/jm00235a007 |
|
Antianaphylactic agents. 4. Synthesis and structure-activity relations of 3-(4-oxo-4H-1-benzopyran-3)acrylic acids, a new series of antiallergic substances, and some related compounds Akira Nohara, Hisashi Kuriki, Taketoshi Saijo, Kiyoshi Ukawa, Tadakazu Murata, Morio Kanno, and Yasushi Sanno pp 34 - 37; DOI: 10.1021/jm00235a008 |
|
Synthesis and absolute stereochemistry of 5-alkyl-5-(3'-hydroxy-1'-methylbutyl)barbituric acid and 5-alkyl-5-(3'-hydroxy-1'-methylbutyl)-2-thiobarbituric acids F. I. Carroll and G. N. Mitchell pp 37 - 41; DOI: 10.1021/jm00235a009 |
|
Aminobenzoic acid diuretics. 7. 3-Substituted 4-phenyl-, 4-arylcarbonyl-, and 4-arylmethyl-5-sulfamoylbenzoic acids and related compounds Ole B. Tvaermose Nielsen, Herta Bruun, Claus Bretting, and Peter W. Feit pp 41 - 50; DOI: 10.1021/jm00235a010 |
|
Antiinflammatory sydnones. 2 John B. Hill, Richard E. Ray, Ray H. Wagner, and Richard L. Aspinall pp 50 - 53; DOI: 10.1021/jm00235a011 |
|
2-Aryl-5-benzoxazolealkanoic acid derivatives with notable antiinflammatory activity David W. Dunwell, Delme Evans, Terrence A. Hicks, Colin H. Cashin, and Ann Kitchen pp 53 - 58; DOI: 10.1021/jm00235a012 |
|
Antitumor agents. 11. Synthesis and cytotoxic activity of epoxides of helenalin related derivatives Kuo-Hsiung Lee, Sun-Hyuk Kim, Hiroshi Furukawa, Claude Piantadosi, and Eng-Shang Huang pp 59 - 63; DOI: 10.1021/jm00235a013 |
|
Preparation and antitumor activity of a rearranged ester of cephalotaxine Kenneth L. Mikolajczak, Richard G. Powell, and Cecil R. Smith pp 63 - 66; DOI: 10.1021/jm00235a014 |
|
Preparation and antileukemic activity of some alkoxybenzo[c]phenanthridinium salts and corresponding dihydro derivatives Robert K. Y. Zee-Cheng and C. C. Cheng pp 66 - 71; DOI: 10.1021/jm00235a015 |
|
Quinuclidine chemistry. 3. .beta.-cis-2-(4'-Chlorobenzhydryl)-3-quinuclidinol, a new central nervous system stimulant. Importance of the benzhydryl configuration E. J. Warawa, N. J. Mueller, and Jonas A. Gylys pp 71 - 74; DOI: 10.1021/jm00235a016 |
|
Pyrido[2,3-d]pyrimidine antibacterial agents. 3. 8-Alkyl- and 8-vinyl-5,8-dihydro-5-oxo-2-(1-piperazinyl)pyrido[2,3-d]pyrimidine-6-carboxylic acids and their derivatives Junichi Matsumoto and Shinsaku Minami pp 74 - 79; DOI: 10.1021/jm00235a017 |
|
Purinylhydantoins. Facile conversion of the naturally occuring N-(purin-6-ylcarbamoyl)-L-amino acids into 3-purin-6-ylhydantoins and 3-cyclohexyl-1-(purin-6-ylcarbamoyl)hydantoins Chung II Hong and Girish B. Chheda pp 79 - 84; DOI: 10.1021/jm00235a018 |
|
Quantitative structure-activity relations for dicoumarol antivitamins K in the uncoupling of mitochondrial oxidative phosphorylation Rosine Labbe-Bois, Claude Laruelle, and Jean J. Godfroid pp 85 - 90; DOI: 10.1021/jm00235a019 |
|
Amidines and related compounds. 6. Structure-activity relations of antihypertensive and antisecretory agents related to clonidine Timothy Jen, Helene Van Hoeven, William Groves, Richard A. McLean, and Bernard Loev pp 90 - 99; DOI: 10.1021/jm00235a020 |
|
Synthesis and biological actions of fragmented derivatives of tetrahydroisoquinolines Duane D. Miller, William V. P. Merritt, Peter F. Kador, and Dennis R. Feller pp 99 - 102; DOI: 10.1021/jm00235a021 |
|
.beta.-Cocaine Robert L. Clarke and Sol J. Daum pp 102 - 104; DOI: 10.1021/jm00235a022 |
|
Synthesis of chlorozotocin, the 2-chloroethyl analog of the anticancer antibiotic streptozotocin Thomas P. Johnston, George S. McCaleb, and John A. Montgomery pp 104 - 106; DOI: 10.1021/jm00235a023 |
|
Synthesis and antimicrobial evaluation of N-D-alanyl-1-aminoethylphosphonic acid Joseph W. Huber, W. Franklin Gilmore, and Larry W. Robertson pp 106 - 108; DOI: 10.1021/jm00235a024 |
|
Centrally acting emetics. 8. Conformational aspects of certain dihydrophenanthrene congeners of apomorphine Joseph G. Cannon, Robert V. Smith, Mohd. A. Aleem, and John Paul Long pp 108 - 110; DOI: 10.1021/jm00235a025 |
|
Centrally acting emetics. 9. Hofmann and Emde degradation products of nuciferine Joseph G. Cannon, Plaston R. Khonje, and John Paul Long pp 110 - 112; DOI: 10.1021/jm00235a026 |
|
Antagonism of slow reacting substance in anaphylaxis (SRS-A) and other spasmogens on the guinea pig tracheal chain by hydratropic acids and their effects on anaphylaxis Margaret E. Greig and Robert L. Griffin pp 112 - 116; DOI: 10.1021/jm00235a027 |
|
Antifertility effects of chlorine-substituted dioxolanes, dithiolanes, and dithianes in male rats Allen F. Hirsch, Kenneth C. Kolwyck, Larry A. Kraft, Roger E. Homm, and Do Won Hahn pp 116 - 117; DOI: 10.1021/jm00235a028 |
|
Triphenylmethane dyes as inhibitors of reverse transcriptase, ribonucleic acid polymerase, and protein synthesis. Structure-activity relations Lon-Lon Liao, Susan B. Horwitz, Mou-Tuan Huang, Arthur P. Grollman, David Steward, and Jack Martin pp 117 - 120; DOI: 10.1021/jm00235a029 |
|
Catechol O-methyltransferase. 5. Structure-activity relations for inhibition by flavonoids Ronald T. Borchardt and Joan A. Huber pp 120 - 122; DOI: 10.1021/jm00235a030 |
|
Book Reviews pp 122 - 122; DOI: 10.1021/jm00235a600 |
|
Somatostatin analogs. Relative importance of the disulfide bridge and of the Ala-Gly side chain for biological activity J. Rivier, P. Brazeau, W. Vale, and R. Guillemin pp 123 - 126; DOI: 10.1021/jm00236a001 |
|
Distal conformation of thyroid hormones. Crystal and molecular structure of 3,5,3'-triiodo-L-thyronine methyl ester Vivian Cody pp 126 - 129; DOI: 10.1021/jm00236a002 |
|
Synthesis and properties of new bradykinin potentiating peptides Mineko Tominaga, John M. Stewart, Therezinha B. Paiva, and Antonio C. M. Paiva pp 130 - 133; DOI: 10.1021/jm00236a003 |
|
Metabolism of carbidopa, (-)-L-.alpha.-hydrazino-3,4-dihydroxy-.alpha.-methylbenzenepropanoic acid monohydrate, in the human, rhesus monkey, dog, and rat Stanley Vickers, Eva K. Stuart, Howard B. Hucker, and William J. A. VandenHeuvel pp 134 - 138; DOI: 10.1021/jm00236a004 |
|
Norepinephrine uptake sites in cardiac tissue. Lack of affinity of 6-hydroxynorepinephrine and related compounds A. Rotman, J. Lundstrom, E. McNeal, J. Daly, and C. R. Creveling pp 138 - 142; DOI: 10.1021/jm00236a005 |
|
Antiarrhythmic agents. 2-, 3-, and 4-Substituted benzylamines David C. Remy, William A. Van Saun, Edward L. Engelhardt, Mary L. Torchiana, and Clement A. Stone pp 142 - 148; DOI: 10.1021/jm00236a006 |
|
Cardioselective .beta.-adrenergic blocking agents. 1. 1-[(3,4-Dimethoxyphenethyl)amino]-3-aryloxy-2-propanols Milton L. Hoefle, Stephen G. Hastings, Robert F. Meyer, Ruth M. Corey, Ann Holmes, and Charlotte D. Stratton pp 148 - 152; DOI: 10.1021/jm00236a007 |
|
Catechol O-methyltransferase. 6. Affinity labeling with N-haloacetyl-3,5-dimethoxy-4-hydroxyphenylalkylamines Ronald T. Borchardt and Dhiren R. Thakker pp 152 - 158; DOI: 10.1021/jm00236a008 |
|
Antiparasitic nitroimidazoles. 8. Derivatives of 2-(4-formylstyryl)-5-nitro-1-vinylimidazole William J. Ross and William B. Jamieson pp 158 - 161; DOI: 10.1021/jm00236a009 |
|
Synthesis and biological evaluation of xanthine oxidase inhibitors. Pyrazolo[3,4-d]pyrimidines and pyrazolo[3,4-b]pyridines Ih Chu and Brian M. Lynch pp 161 - 165; DOI: 10.1021/jm00236a010 |
|
Synthesis and biological activity of some ethers of testosterone. Implications concerning the biological activity of esters of testosterone Alan J. Solo, Natalie Bejba, Peter Hebborn, and Marian May pp 165 - 168; DOI: 10.1021/jm00236a011 |
|
Substituted pyrazolo corticoids as topical antiinflammatory agents John Hannah, Kenneth Kelly, Arthur A. Patchett, Sanford L. Steelman, and Evan R. Morgan pp 168 - 172; DOI: 10.1021/jm00236a012 |
|
Preparation, hydrolysis, and oral absorption of .alpha.-carboxy esters of carbenicillin J. Peter Clayton, Martin Cole, Stephen W. Elson, Kenneth D. Hardy, Linda W. Mizen, and Robert Sutherland pp 172 - 177; DOI: 10.1021/jm00236a013 |
|
5-Aryl-2,3-dihydro-5H-imidazo[2,1-a]isoindol-5-ols. Novel class of anorectic agents Paul Aeberli, Phillip Eden, John H. Gogerty, William J. Houlihan, and Chris Penberthy pp 177 - 182; DOI: 10.1021/jm00236a014 |
|
Anorectic agents. 2. Structural analogs of 5-(p-chlorophenyl)-2,3-dihydro-5H-imidazo[2,1-a]isoindol-5-ol Paul Aeberli, Phillip Eden, John H. Gogerty, William J. Houlihan, and Chris Penberthy pp 182 - 185; DOI: 10.1021/jm00236a015 |
|
Neuroleptic agents of the benzocycloheptapyridoisoquinoline series. 1. Syntheses and stereochemical and structural requirements for activity of butaclamol and related compounds Francois T. Bruderlein, Leslie G. Humber, and Katherine Voith pp 185 - 188; DOI: 10.1021/jm00236a016 |
|
Chemistry and antiinflammatory activities of prodolic acid and related 1,3,4,9-tetrahydropyrano[3,4-b]indole-1-alkanoic acids. 1 Christopher A. Demerson, Leslie G. Humber, Thomas A. Dobson, and Rene R. Martel pp 189 - 191; DOI: 10.1021/jm00236a017 |
|
Synthesis of thieno[2,3-b]azepin-4-ones as potential antineoplastic agents R. F. Koebel, L. L. Needham, and C. De Witt Blanton pp 192 - 194; DOI: 10.1021/jm00236a018 |
|
Synthesis of bis(aziridinyl)phosphinyl-N-hydroxyurethane derivatives as antineoplastic agents Y. Y. Hsiao, T. J. Bardos, G. L. Wampler, and W. Regelson pp 195 - 198; DOI: 10.1021/jm00236a019 |
|
Vulpinic acids as potential antiinflammatory agents. 1. Vulpinic acids with substituents in the aromatic rings F. R. Foden, J. McCormick, and D. M. O'Mant pp 199 - 203; DOI: 10.1021/jm00236a020 |
|
Hydroaromatic analogs of 2-nitro-1,3-indandiones Derek R. Buckle, Neil J. Morgan, and Harry Smith pp 203 - 206; DOI: 10.1021/jm00236a021 |
|
1,5-Ethano-2,3,4,5-tetrahydro-1H-3-benzazepines Lewis A. Walter and Wei K. Chang pp 206 - 208; DOI: 10.1021/jm00236a022 |
|
Correlation of psychotomimetic activity of phenethylamines and amphetamines with 1-octanol-water partition coefficients C. F. Barfknecht, David E. Nichols, and W. J. Dunn pp 208 - 210; DOI: 10.1021/jm00236a023 |
|
.beta.-Adrenergic blockade by 3-[3-(substituted amino)-2-hydroxypropoxy]-5-hydroxybenzyl alcohols Charles F. Schwender, Russell E. Pike, John Shavel, and Harvey R. Kaplan pp 211 - 213; DOI: 10.1021/jm00236a024 |
|
Hashish. Importance of the phenolic hydroxyl group in tetrahydrocannabinols D. B. Uliss, H. C. Dalzell, G. R. Handrick, J. F. Howes, and R. K. Razdan pp 213 - 215; DOI: 10.1021/jm00236a025 |
|
Stereoselective synthetic route to (R)-zearalanone C. Allan Peters and Richard N. Hurd pp 215 - 217; DOI: 10.1021/jm00236a026 |
|
Synthesis and biological properties of 17.alpha.-furylestradiol and dihydroequilin derivatives Clara Revesz and Yvon Lefebvre pp 217 - 219; DOI: 10.1021/jm00236a027 |
|
Synthesis and estrogenic properties of 7.alpha.,8.alpha.-epoxy- and 7.alpha.,8.alpha.-methyleneestradiols Yvon Lefebvre, David J. Marshall, and Clara Revesz pp 220 - 222; DOI: 10.1021/jm00236a028 |
|
Quinazolines and 1,4-benzodiazepines. 67. 5-Ferrocenyl-1,4-benzodiazepin-2-ones Robert Kalish, Thomas V. Steppe, and Armin Walser pp 222 - 224; DOI: 10.1021/jm00236a029 |
|
6-Methyl-1,2,3,5-tetrahydroimidazo[2,1-b]quinazolin-2-one, a potent inhibitor of ADP-induced platelet aggregation W. N. Beverung and R. A. Partyka pp 224 - 225; DOI: 10.1021/jm00236a030 |
|
(1-Oxo-2-substituted-5-indanyloxy)acetic acids, a new class of potent renal agents possessing both uricosuric and saluretic activity. Reexamination of the role of sulfhydryl binding in the mode of action of acylphenoxyacetic acid saluretics E. J. Cragoe, E. M. Schultz, J. D. Schneeberg, G. E. Stokker, O. W. Woltersdorf, G. M. Fanelli, and L. S. Watson pp 225 - 228; DOI: 10.1021/jm00236a031 |
|
Book Reviews pp 228 - 230; DOI: 10.1021/jm00236a600 |
|
Relations between the biological and physicochemical properties of series of compounds Richard M. Hyde pp 231 - 233; DOI: 10.1021/jm00237a001 |
|
Application of regression analysis to the hypoglycemic activities of a series of substituted benzenesulfonamidopyrimidines Joachim K. Seydel, Hanns Ahrens, and Wolfgang Losert pp 234 - 240; DOI: 10.1021/jm00237a002 |
|
Homologous N-alkylnorketobemidones. Correlation of receptor binding with analgesic potency Raymond S. Wilson, Michael E. Rogers, Candace B. Pert, and Soloman H. Snyder pp 240 - 242; DOI: 10.1021/jm00237a003 |
|
Hypocholesteremic derivatives of styrylacetic acid. 1. gem-Dimethyl analogs of benzalbutyric acid Eugene S. Stratford pp 242 - 245; DOI: 10.1021/jm00237a004 |
|
Antiviral quinolinehydrazones. Modified Free-Wilson analysis Jean Thomas, Charles E. Berkoff, Walter B. Flagg, John J. Gallo, Richard F. Haff, Carl A. Pinto, Cesare Pellerano, and Luisa Savini pp 245 - 250; DOI: 10.1021/jm00237a005 |
|
Preparation and anticoagulant activity of trimethylsilyl heparin in Carbowax Edward E. Nishizawa, Daniel J. Wynalda, Robert E. Harmon, Kalyan K. De, and Surendra K. Gupta pp 250 - 253; DOI: 10.1021/jm00237a006 |
|
Chemotherapeutic nitroheterocycles. 18. 2-(5-Nitro-2-imidazolylmethylene)-1-indanones, -1-tetralones, and -acetophenones substituted by aminoalkoxy groups C. Rufer, H. J. Kessler, and E. Schroeder pp 253 - 258; DOI: 10.1021/jm00237a007 |
|
Narcotic antagonists. 4. Carbon-6 derivatives of N-substituted noroxymorphones as narcotic antagonists Elliot F. Hahn, Jack Fishman, and Richard D. Heilman pp 259 - 262; DOI: 10.1021/jm00237a008 |
|
Synthesis and evaluation of 6-arylacetamido-2,4-diaminoquinazolines and related compounds as folic acid antagonists John B. Hynes and Wallace T. Ashton pp 263 - 265; DOI: 10.1021/jm00237a009 |
|
Synthesis of a new metabolite of acetylmethadol Richard N. Booher and Albert Pohland pp 266 - 268; DOI: 10.1021/jm00237a010 |
|
Synthesis of 15-keto-6.beta.,7.beta.-methyleneprogesterone. Effect of the 6.beta.,7.beta.-methylene group on mineralocorticoid activity Leland J. Chinn and Bipin N. Desai pp 268 - 271; DOI: 10.1021/jm00237a011 |
|
Synthesis and antifolate activity of new diaminopyrimidines and diaminopurines in enzymic and cellular systems Ivan Kavai, Lawrence H. Mead, Jadwiga Drobniak, and Sigmund F. Zakrzewski pp 272 - 275; DOI: 10.1021/jm00237a012 |
|
Synthesis and biological activity of LH-RH analogs modified at the carboxyl terminus David H. Coy, Esther J. Coy, Andrew V. Schally, and Jesus A. Vilchez-Martinez pp 275 - 277; DOI: 10.1021/jm00237a013 |
|
Fibrin-stabilizing factor inhibitors. 12. 5-Dibenzylaminopentylamine and related compounds, a new type of FSF [fibrin-stabilizing factor] inhibitors Kurt Juergen Hoffmann, Pal Stenberg, Christine Ljunggren, Uno Svensson, J. Lars G. Nilsson, Olle Eriksson, Ann Hartkoorn, and Ragnar Lunden pp 278 - 284; DOI: 10.1021/jm00237a014 |
|
[1-.beta.-Mercapto-.beta.,.beta.-pentamethylenepropionic acid]oxytocin, a potent inhibitor of oxytocin John J. Nestor, Martha F. Ferger, and Vincent Du Vigneaud pp 284 - 287; DOI: 10.1021/jm00237a015 |
|
Synthesis of isoesteres of p-amidinophenylpyruvic acid. Inhibitors of trypsin, thrombin, and pancreatic kallikrein Larry J. Loeffler, Eng-Chun Mar, J. D. Geratz, and Lynda B. Fox pp 287 - 292; DOI: 10.1021/jm00237a016 |
|
Base-catalyzed and cholinesterase-catalyzed hydrolysis of acetylcholine and optically active analogs Katharine B. Schowen, Edward E. Smissman, and William F. Stephen pp 292 - 300; DOI: 10.1021/jm00237a017 |
|
Potential inhibitors of S-adenosylmethionine-dependent methyltransferases. 3. Modifications of the sugar portion of S-adenosylhomocysteine Ronald T. Borchardt and Yih Shiong Wu pp 300 - 304; DOI: 10.1021/jm00237a018 |
|
Norepinephrine N-methyltransferase inhibition by benzamidines, phenylacetamidines, benzylguanidines, and phenylethylguanidines Ray W. Fuller, Betty W. Roush, Harold D. Snoddy, William A. Day, and Bryan B. Molloy pp 304 - 307; DOI: 10.1021/jm00237a019 |
|
Structure and stereochemistry of some 1,2-disubstituted mitosenes from solvolysis of mitomycin C and Mitomycin A Wesley G. Taylor and William A. Remers pp 307 - 311; DOI: 10.1021/jm00237a020 |
|
Synthesis and antitrichomonal activity of certain pyrazolo[1,5-a]pyrimidines Keitaro Senga, Thomas Novinson, Robert H. Springer, Ravindra P. Rao, Darrell E. O'Brien, Roland K. Robins, and Henry R. Wilson pp 312 - 314; DOI: 10.1021/jm00237a021 |
|
3-Substituted 2',3'-dihydroestra-1,3,5(10)-trieno[16.alpha.,17.alpha.-b]furan-17.beta.-ols as potential estrogens Alan Dinner, Rafik H. Bishara, and Bonnie S. Rutherford pp 314 - 315; DOI: 10.1021/jm00237a022 |
|
Hypotensive activity of 3-alkyl-2-iminobenzothiazolines Stephen W. Horgan, James K. Woodward, Alfred Richardson, and Albert A. Carr pp 315 - 318; DOI: 10.1021/jm00237a023 |
|
Etonitazene. Improved synthesis Frank I. Carroll and Michael C. Coleman pp 318 - 320; DOI: 10.1021/jm00237a024 |
|
Preparation of a new immunosuppressant, 4,5-bis(aminomethyl)acridine F. K. Hess and P. B. Stewart pp 320 - 321; DOI: 10.1021/jm00237a025 |
|
Book Reviews pp 321 - 322; DOI: 10.1021/jm00237a600 |
|
Radioprotective stereostructure-activity study of cis- and trans-2-mercaptocyclobutylamine analogs and homologs of 2-mercaptoethylamine Ronald W. Hart, Ruth E. Gibson, J. Donald Chapman, Antoon P. Reuvers, Birandra K. Sinha, Robert K. Griffith, and Donald T. Witiak pp 323 - 331; DOI: 10.1021/jm00238a001 |
|
Structure-activity correlations among rifamycin B amides and hydrazides Frank R. Quinn, John S. Driscoll, and Corwin Hansch pp 332 - 339; DOI: 10.1021/jm00238a002 |
|
Nucleic acids. 14. ara-Cytidine acylates. Use of drug design predictors in structure-activity relation correlation W. J. Wechter, M. A. Johnson, C. M. Hall, D. T. Warner, A. E. Berger, A. H. Wenzel, D. T. Gish, and G. L. Neil pp 339 - 344; DOI: 10.1021/jm00238a003 |
|
Linear regression analysis of inhibitory potency of organic disulfides against Histoplasma capsulatum L. J. Schaad, R. H. Werner, Lynn Dillon, Lamar Field, and C. Emory Tate pp 344 - 351; DOI: 10.1021/jm00238a004 |
|
Substituted thiadiazolines as inhibitors of central nervous system carbonic anhydrase James J. Lukes and Karl A. Nieforth pp 351 - 354; DOI: 10.1021/jm00238a005 |
|
Potential inhibitors of L-asparagine biosynthesis. 2. Chemistry and biological activity of .beta.-hydroxyaspartic acid and its derivatives Michael Mokotoff, James F. Bagaglio, and Bharat S. Parikh pp 354 - 358; DOI: 10.1021/jm00238a006 |
|
Prostaglandins and congeners. 7. Synthesis of simplified prostaglandins. Inhibition of gastric acid secretion by 2-(.omega.-carboxyalkyl)-3-alkylcycloalkanones John F. Poletto, Karel F. Bernady, David Kupfer, Ruth Partridge, and Martin J. Weiss pp 359 - 362; DOI: 10.1021/jm00238a007 |
|
Synthesis and pharmacology of some 2-aminotetralins. Dopamine receptor agonists John D. McDermed, Gerald M. McKenzie, and Arthur P. Phillips pp 362 - 367; DOI: 10.1021/jm00238a008 |
|
Potential antitumor agents. 12. 2-Formyl-4-aminophenylpyridine thiosemicarbazones Krishna C. Agrawal, Barbara A. Booth, Suzanne M. DeNuzzo, and Alan C. Sartorelli pp 368 - 371; DOI: 10.1021/jm00238a009 |
|
Synthesis and tumor-uptake study of phosphate esters of polyhedral hydroxyboranes Rebecca A. Bechtold, A. Kaczmarczyk, and Janette R. Messer pp 371 - 376; DOI: 10.1021/jm00238a010 |
|
Cyclophosphamide metabolites and their related compounds. 2. Preparation of an active species of cyclophosphamide and related compounds Akira Takamizawa, Saichi Matsumoto, Tsuyoshi Iwata, Yoshihiro Tochino, Ken Katagiri, Kenji Yamaguchi, and Osamu Shiratori pp 376 - 383; DOI: 10.1021/jm00238a011 |
|
Anticonvulsants. 5. Derivatives of 5-ethyl-5-phenylhydantoin and 5,5-diphenylhydantoin Julius A. Vida, Mary H. O'Dea, Carlos M. Samour, and John F. Reinhard pp 383 - 385; DOI: 10.1021/jm00238a012 |
|
Antiinflammatory fluoroalkanesulfonanilides. 3. Other fluoroalkanesulfonamido diaryl systems G. G. I. Moore, J. K. Harrington, and K. F. Swingle pp 386 - 391; DOI: 10.1021/jm00238a013 |
|
Antiallergic activity of 4-hydroxy-3-nitrocoumarins Derek R. Buckle, Barrie C. C. Cantello, Harry Smith, and Barbara A. Spicer pp 391 - 394; DOI: 10.1021/jm00238a014 |
|
Cyclopenta[f]isoquinoline derivatives designed to bind specifically to native deoxyribonucleic acid. 1. Synthesis of 3-ethoxy-8-methyl-7(5)H-cyclopenta[f]isoquinoline Nitya G. Kundu, John A. Wright, Kato L. Perlman, William Hallett, and Charles Heidelberger pp 395 - 399; DOI: 10.1021/jm00238a015 |
|
Cyclopenta[f]isoquinoline derivatives designed to bind specifically to native deoxyribonucleic acid. 2. Synthesis of 6-carbamylmethyl-8-methyl-7(5)H-cyclopenta[f]isoquinolin-3(2H)-one and its interaction with deoxyribonucleic acids and poly(deoxyribonucleotides) Nitya G. Kundu, William Hallett, and Charles Heidelberger pp 399 - 403; DOI: 10.1021/jm00238a016 |
|
Chemistry of cephalosporin antibiotics. 30. 3-Methoxy- and 3-halo-3-cephems Robert R. Chauvette and Pamela A. Pennington pp 403 - 408; DOI: 10.1021/jm00238a017 |
|
Electronic structures of cephalosporins and penicillins. 4. Modeling acylation by the .beta.-lactam ring Donald B. Boyd, Robert B. Hermann, David E. Presti, and Max M. Marsh pp 408 - 417; DOI: 10.1021/jm00238a018 |
|
Pseudosymmetry in the structure of luteinizing hormone-releasing hormone. Series of novel analogs Christopher R. Beddell, Peter J. Fraser, David Gilbert, Peter J. Goodford, Lawrence A. Lowe, and Samuel Wilkinson pp 417 - 423; DOI: 10.1021/jm00238a019 |
|
Adrenocorticotropin. 47. Synthesis and biological activity of adrenocorticotropic peptides modified at the tryptophan position James Blake and Choh Hao Li pp 423 - 426; DOI: 10.1021/jm00238a020 |
|
Isotope effects in enzymic N-demethylation of tertiary amines Mahmoud M. Abdel-Monem pp 427 - 430; DOI: 10.1021/jm00238a021 |
|
Antiparasitic nitroimidazoles. 9. Synthesis of some 2-(4-dialkylaminomethylstyryl)- and 2-(4-amidinostyryl)-5-nitro-1-vinylimidazoles William J. Ross and William B. Jamieson pp 430 - 432; DOI: 10.1021/jm00238a022 |
|
Cycloalkanones. 6. Separation of hypocholesterolemic and antifertility activities in derivatives of 2,8-dibenzylcyclooctanone G. L. Carlson, I. H. Hall, and C. Piantadosi pp 432 - 434; DOI: 10.1021/jm00238a023 |
|
Homologs of dopa, .alpha.-methyldopa, and dopamine as potential cardiovascular drugs M. Winn, R. Rasmussen, F. Minard, J. Kyncl, and N. Plotnikoff pp 434 - 437; DOI: 10.1021/jm00238a024 |
|
N-Cyclopropyltryptamines, potent monoamine oxidase inhibitors M. Winn, B. W. Horrom, R. R. Rasmussen, E. B. Chappell, and N. P. Plotnikoff pp 437 - 438; DOI: 10.1021/jm00238a025 |
|
Synthesis of 8-(3'-deoxy-.alpha.-D-threo-pentofuranosyl)adenine and 9-(3'-deoxy-.alpha.-D-threo-pentofuranosyl)adenine Hassan S. El Khadem and Thakur D. Audichya pp 438 - 441; DOI: 10.1021/jm00238a026 |
|
.beta.-Aminocinnamonitriles as potential antiinflammatory agents S. A. Lang and E. Cohen pp 441 - 443; DOI: 10.1021/jm00238a027 |
|
Book Reviews pp 444 - 446; DOI: 10.1021/jm00238a600 |
|
Synthesis and biological evaluation of some 10-substituted 2,3-dihydroimidazo[2,1-b]quinazolin-5(10H)-ones, a new class of bronchodilators Goetz E. Hardtmann, Gabor Koletar, Oskar R. Pfister, John H. Gogerty, and Louis C. Iorio pp 447 - 453; DOI: 10.1021/jm00239a001 |
|
Synthesis and biological evaluation of fragmented derivatives of tetrahydroisoquinolines. 2. Trimetoquinol studies Duane D. Miller, Peter Osei-Gyimah, John Bardin, and Dennis R. Feller pp 454 - 457; DOI: 10.1021/jm00239a002 |
|
Porphyria-inducing activity of a series of pyridine and dihydropyridine compounds. Investigation in a cell culture system M. W. Roomi pp 457 - 460; DOI: 10.1021/jm00239a003 |
|
Adenosine cyclic 3',5'-monophosphate phosphodiesterase inhibitors. 2. 3-Substituted 5,7-dialkylpyrazolo[1,5-a]pyrimidines Thomas Novinson, Jon P. Miller, Mieka Scholten, Roland K. Robins, Lionel N. Simon, Darrell E. O'Brien, and Rich B. Meyer pp 460 - 464; DOI: 10.1021/jm00239a004 |
|
Synthesis and antitumor activity of 5'-phosphates and cyclic 3',5'-phosphates derived from biologically active nucleosides Chung Il Hong, George L. Tritsch, Arnold Mittelman, Peter Hebborn, and Girish B. Chheda pp 465 - 473; DOI: 10.1021/jm00239a005 |
|
Synthesis and biological activity of 4-(.beta.-D-ribofuranosyl)-1,3-dihydroxybenzene (1,3-dideazauridine) R. A. Sharma, M. Bobek, and A. Bloch pp 473 - 476; DOI: 10.1021/jm00239a006 |
|
New aromatic diamidines with central .alpha.-oxyalkane or .alpha.,.omega.-dioxyalkane chains. Structure-activity relations for the inhibition of trypsin, pancreatic kallikrein, and thrombin and for the inhibition of the overall coagulation process J. D. Geratz, M. C. F. Cheng, and R. R. Tidwell pp 477 - 481; DOI: 10.1021/jm00239a007 |
|
Synthesis and study of glutaryl-S-(.omega.-aminoalkyl)-L-cysteinylglycines as inhibitors of glyoxalase I G. W. Phillips and S. J. Norton pp 482 - 486; DOI: 10.1021/jm00239a008 |
|
Preparation and properties of 5-phenylphenoxymethylpenicillin Hubert Vanderhaeghe and Jozef Thomis pp 486 - 490; DOI: 10.1021/jm00239a009 |
|
Stereospecific synthesis of the 6.beta.-hydroxy metabolites of naltrexone and naloxone Nithiananda Chatterjie, Charles E. Inturrisi, Hyman B. Dayton, and Harold Blumberg pp 490 - 492; DOI: 10.1021/jm00239a010 |
|
Synthesis of N10-methyl-4-thiofolic acid and related compounds Robert D. Elliott, Carroll Temple, Jerry L. Frye, and John A. Montgomery pp 492 - 496; DOI: 10.1021/jm00239a011 |
|
Analgesic activity of the epimeric tropane analogs of meperidine. Physical and pharmacological study Sol J. Daum, Catherine M. Martini, Rudolph K. Kullnig, and Robert L. Clarke pp 496 - 501; DOI: 10.1021/jm00239a012 |
|
Probiotics. Antistaphylococcal and antifibrinolytic activities of .omega.-amino- and .omega.-guanidinoalkanesulfonic acids Akira Fujii and Elton S. Cook pp 502 - 505; DOI: 10.1021/jm00239a013 |
|
Carbon-13 magnetic resonance spectroscopy of drugs. Sulfonamides Ching Jer Chang, Heinz G. Floss, and Garnet E. Peck pp 505 - 509; DOI: 10.1021/jm00239a014 |
|
Antiinflammatory .beta.-arylamidoacrylic acids Robert T. Buckler, Harold E. Hartzler, and Barrie M. Phillips pp 509 - 513; DOI: 10.1021/jm00239a015 |
|
Synthesis and thin-layer chromatographic, ultraviolet, and mass spectral properties of the anticoagulant phenprocoumon and its monohydroxylated derivatives Lance R. Pohl, Rodney Haddock, William A. Garland, and William F. Trager pp 513 - 519; DOI: 10.1021/jm00239a016 |
|
Biotransformation of phenprocoumon in the rat Rodney E. Haddock, William F. Trager, and Lance R. Pohl pp 519 - 523; DOI: 10.1021/jm00239a017 |
|
Potential antimalarials. 9. Resolution of .alpha.-diheptylaminomethyl-6-bromo-9-phenanthrenemethanol by an unusual method D. E. Pearson and Adam A. Rosenberg pp 523 - 524; DOI: 10.1021/jm00239a018 |
|
Substituted 1-[(5-nitrofurfurylidene)amino]-4-imidazolin-2-ones Harry R. Snyder and Raymond Freedman pp 524 - 526; DOI: 10.1021/jm00239a019 |
|
Synthesis of a fluorescent derivative of amethopterin G. R. Gapski, J. M. Whiteley, J. I. Rader, P. L. Cramer, G. B. Hendersen, V. Neef, and F. M. Huennekens pp 526 - 528; DOI: 10.1021/jm00239a020 |
|
Inhibition of phenylalanyl-tRNA synthetase by aromatic guanidines and amidines Peter V. Danenberg and Daniel V. Santi pp 528 - 530; DOI: 10.1021/jm00239a021 |
|
2-Phenethylimidazole derivatives. Synthesis and antimycotic properties Erik F. Godefroi, Jack J. H. Geenen, Bert Van Klingeren, and Leo J. Van Wijngaarden pp 530 - 533; DOI: 10.1021/jm00239a022 |
|
Preparation of fluorine-18-labeled haloperidol C. S. Kook, M. F. Reed, and G. A. Digenis pp 533 - 535; DOI: 10.1021/jm00239a023 |
|
Analogs of camptothecin James A. Bristol, Daniel L. Comins, Richard W. Davenport, Michael J. Kane, Robert E. Lyle, John R. Maloney, David E. Portlock, and Susan B. Horwitz pp 535 - 537; DOI: 10.1021/jm00239a024 |
|
Book Reviews pp 537 - 538; DOI: 10.1021/jm00239a600 |
|
Pattern recognition and structure-activity relation studies. Computer-assisted prediction of antitumor activity in structurally diverse drugs in an experimental mouse brain tumor system K. C. Chu, R. J. Feldmann, M. B. Shapiro, G. F. Hazard, and R. I. Geran pp 539 - 545; DOI: 10.1021/jm00240a001 |
|
Partition coefficients and the structure-activity relation of the anesthetic gases Corwin Hansch, Antonio Vittoria, Carlo Silipo, and Priscilla Y. Jow pp 546 - 548; DOI: 10.1021/jm00240a002 |
|
Liquid-liquid partition coefficients by high-pressure liquid chromatography John M. McCall pp 549 - 552; DOI: 10.1021/jm00240a003 |
|
Synthesis and pharmacological properties of 4-piperazino-5-methylthiopyrimidines. Selection of new antiemetic agents Georges Mattioda, Pierre Obellianne, Henri Gauthier, Gerard Loiseau, Rene Millischer, Anne M. Donadieu, and Michel Mestre pp 553 - 559; DOI: 10.1021/jm00240a004 |
|
Synthesis and biological activity of some 8-substituted selenoguanosine cyclic 3',5'-phosphates and related compounds Shih Hsi Chu, Chyng Yann Shiue, and Ming Yu Chu pp 559 - 564; DOI: 10.1021/jm00240a005 |
|
Nucleosides of 2-azapurines. 7H-Imidazo[4,5-d]-1,2,3-triazines. 2 John A. Montgomery, Anne G. Laseter, Anita T. Shortnacy, Sarah J. Clayton, and H. Jeanette Thomas pp 564 - 567; DOI: 10.1021/jm00240a006 |
|
Decomposition of N-(2-chloroethyl)-N-nitrosoureas in aqueous media John A. Montgomery, Ruby James, George S. McCaleb, Marion C. Kirk, and Thomas P. Johnston pp 568 - 571; DOI: 10.1021/jm00240a007 |
|
2-Halo derivatives of 3'-acetamido-3'-deoxyadenosine John A. Montgomery, Kathleen Hewson, and Anne G. Laseter pp 571 - 573; DOI: 10.1021/jm00240a008 |
|
2-Aryloxymethyl-2,3,5,6-tetrahydro-1,4-oxazines, a new class of antidepressants David T. Greenwood, Keith B. Mallion, Alexander H. Todd, and Ralph W. Turner pp 573 - 577; DOI: 10.1021/jm00240a009 |
|
3,4-Dihydro-1H-1,4-oxazino[4,3-a]indoles as potential antidepressants Christopher A. Demerson, George Santroch, Leslie G. Humber, and Marie P. Charest pp 577 - 580; DOI: 10.1021/jm00240a010 |
|
Oxidation of furans. 3. Estrogenic properties of lactones and anhydrides derived from the oxidation of 17.alpha.-[3-furyl]estradiol derivatives Yvon Lefebvre and Clara Revesz pp 581 - 583; DOI: 10.1021/jm00240a011 |
|
Synthesis and antiinflammatory activity of some 1,6-methano[10]annuleneacetic acids P. H. Nelson, G. A. Bartsch, K. G. Untch, and J. H. Fried pp 583 - 586; DOI: 10.1021/jm00240a012 |
|
Quinuclidine chemistry. 4. Diuretic properties of cis-3-amino-2-benzhydrylquinuclidine E. J. Warawa, N. J. Mueller, and J. Stuart Fleming pp 587 - 593; DOI: 10.1021/jm00240a013 |
|
Butyrophenones as hypotensive agents. Derivatives of 4-aryl-4-(hydroxymethyl)cyclohexylamine Daniel Lednicer, D. Edward Emmert, Alan D. Rudzik, and Boyd E. Graham pp 593 - 599; DOI: 10.1021/jm00240a014 |
|
Potential inhibitors of polyamine biosynthesis. 2. .alpha.-Alkyl- and benzyl-(+-)-ornithine Mohmoud M. Abdel-Monem, Nancy E. Newton, Bartholomeus C. Ho, and Charles E. Weeks pp 600 - 604; DOI: 10.1021/jm00240a015 |
|
Physicochemical-activity relations in practice. 1. Rational and self-consistent data bank Franklin E. Norrington, Richard M. Hyde, Stanley G. Williams, and Raymond Wootton pp 604 - 607; DOI: 10.1021/jm00240a016 |
|
Physicochemical-activity relations in practice. 2. Rational selection of benzenoid substituents Raymond Wootton, Robert Cranfield, G. Clive Sheppey, and Peter J. Goodford pp 607 - 613; DOI: 10.1021/jm00240a017 |
|
Synthesis and biological activity of luteinizing hormone-releasing hormone and related peptides Derek J. Schafer, Alan D. Black, John D. Bower, and D. Barry Crighton pp 613 - 619; DOI: 10.1021/jm00240a018 |
|
Effect of 9-hydroxylation on benzomorphan antagonist activity Noel F. Albertson pp 619 - 621; DOI: 10.1021/jm00240a019 |
|
Quantitative structure-activity relations in the .DELTA.6-6-substituted progesterone series. Reappraisal John G. Topliss and Elliot L. Shapiro pp 621 - 623; DOI: 10.1021/jm00240a020 |
|
4-Amino-5-arylpyrimidines as antiinflammatory agents S. A. Lang and E. Cohen pp 623 - 625; DOI: 10.1021/jm00240a021 |
|
Monocyclic antibiotic .beta.-lactams Riaz F. Abdulla and Kenneth H. Fuhr pp 625 - 627; DOI: 10.1021/jm00240a022 |
|
7-N-Amidinocephalosporins J. Altman, E. Karoly, and N. Maoz pp 627 - 630; DOI: 10.1021/jm00240a023 |
|
Synthesis of .alpha.-1-noracetylmethadol. Facile N-demethylation of .alpha.-1-acetylmethadol Nithiananda Chatterjie and Charles E. Inturrisi pp 630 - 631; DOI: 10.1021/jm00240a024 |
|
Synthesis of quinazoline analogs of isofolic acid John B. Hynes and Claudia M. Garrett pp 632 - 634; DOI: 10.1021/jm00240a025 |
|
Synthesis and biologic evaluation of major metabolites of N-(2-chloroethyl)-N'-cyclohexyl-N-nitrosourea Thomas P. Johnston, George S. McCaleb, and John A. Montgomery pp 634 - 637; DOI: 10.1021/jm00240a026 |
|
3-Substituted 2-formylquinoxaline 1,4-dioxides M. L. Edwards, R. E. Bambury, and H. W. Ritter pp 637 - 639; DOI: 10.1021/jm00240a027 |
|
Hydroxylated 2,3,4,9-tetrahydro-1H-carbazol-3-amines. New class of experimental cardiotonic drugs Aram Mooradian, Allan G. Hlavac, Paul E. Dupont, Malcolm R. Bell, and Adawia A. Alousi pp 640 - 641; DOI: 10.1021/jm00240a028 |
|
Book Reviews pp 641 - 646; DOI: 10.1021/jm00240a600 |
|
Microelectrometric titration measurement of the pKa's and partition and drug distribution coefficients of narcotics and narcotic antagonists and their pH and temperature dependence Joyce J. Kaufman, Nora M. Semo, and Walter S. Koski pp 647 - 655; DOI: 10.1021/jm00241a001 |
|
Quantum chemical studies of morphine-like opiate narcotics. Effect of N-substituent variations Gilda H. Loew and Donald S. Berkowitz pp 656 - 662; DOI: 10.1021/jm00241a002 |
|
Conformation of histamine derivatives. 5. Molecular orbital calculation of the H1-receptor essential conformation of histamine L. Farnell, W. G. Richards, and C. R. Ganellin pp 662 - 666; DOI: 10.1021/jm00241a003 |
|
Tricyclic quinuclidylidenes as potential antihistamine-bronchodilating agents Frank J. Villani, Thomas A. Mann, and Elizabeth A. Wefer pp 666 - 669; DOI: 10.1021/jm00241a004 |
|
Synthesis and biological activity of spin-labeled analogs of biotin, hexamethonium, decamethonium, dichlorisoproterenol, and propranolol Birandra K. Sinha and Colin F. Chignell pp 669 - 673; DOI: 10.1021/jm00241a005 |
|
Adrenergic agents. 3. Synthesis and adrenergic activity of some catecholamine analogs bearing a substituted sulfonyl or sulfonylalkyl group in the meta position Carl Kaiser, Mark S. Schwartz, Donald F. Colella, and Joe R. Wardell pp 674 - 683; DOI: 10.1021/jm00241a006 |
|
N-Hydroxylation of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane by rabbit liver microsomes J. Gal, L. D. Gruenke, and N. Castagnoli pp 683 - 688; DOI: 10.1021/jm00241a007 |
|
Triarylpyridylethanols and triarylpyridylethylenes. Chemistry and antifertility effects Alfred Richardson, Jasti B. Choudary, and Dorsey E. Holtkamp pp 689 - 691; DOI: 10.1021/jm00241a008 |
|
Synthesis and antiinflammatory activity of some 2-substituted .alpha.-methyl-5-benzimidazoleacetic acids David W. Dunwell, Delme Evans, Christine E. Smith, and W. R. Nigel Williamson pp 692 - 694; DOI: 10.1021/jm00241a009 |
|
Analgesics. 3. Selected 1-substituted and 1,3-disubstituted 5-propionoxy-5-(1-phenylethyl)barbituric acids Julius A. Vida, Carlos M. Samour, Mary H. O'Dea, and John F. Reinhard pp 694 - 696; DOI: 10.1021/jm00241a010 |
|
Hydrogenated benzo[f]quinolines and benz[e]indoles as analgetics. 1 Mikio Takeda, Mikihiko Konda, Yasushi Honma, Hirozumi Inoue, Seiichi Saito, Hiroshi Kugita, Seiichi Nurimoto, and Goro Hayashi pp 697 - 699; DOI: 10.1021/jm00241a011 |
|
Analgesic properties of the tetrahydrocannabinols, their metabolites, and analogs Raymond S. Wilson and Everette L. May pp 700 - 703; DOI: 10.1021/jm00241a012 |
|
Synthesis and antitumor properties of new glycosides of daunomycinone and adriamycinone Federico Arcamone, Sergio Penco, Aristide Vigevani, Silvio Redaelli, Giuliano Franchi, Aurelio Di Marco, Anna M. Casazza, Teresa Dasdia, Franca Formelli, and et al. pp 703 - 707; DOI: 10.1021/jm00241a013 |
|
Synthesis and biological activity of some antitumor benzophenanthridinium salts Frank R. Stermitz, John P. Gillespie, Luis G. Amoros, Raquel Romero, Thomas A. Stermitz, Kenneth A. Larson, Steven Earl, and James E. Ogg pp 708 - 713; DOI: 10.1021/jm00241a014 |
|
Biologically active polycycloalkanes. 1. Antiviral adamantane derivatives Koji Aigami, Yoshiaki Inamoto, Naotake Takaishi, Kenichi Hattori, Akira Takatsuki, and Gakuzo Tamura pp 713 - 721; DOI: 10.1021/jm00241a015 |
|
Synthesis and antiviral activity of certain 5'-monophosphates of 9-D-arabinofuranosyladenine and 9-D-arabinofuranosylhypoxanthine Ganapathi R. Revankar, John H. Huffman, Lois B. Allen, Robert W. Sidwell, Roland K. Robins, and Richard L. Tolman pp 721 - 726; DOI: 10.1021/jm00241a016 |
|
4-Hydroxy-3-nitro-2-quinolones and related compounds as inhibitors of allergic reactions Derek R. Buckle, Barrie C. C. Cantello, Harry Smith, and Barbara A. Spicer pp 726 - 732; DOI: 10.1021/jm00241a017 |
|
Antiallergic activity of .omega.-nitroacetophenones Derek R. Buckle, Barrie C. C. Cantello, Neil J. Morgan, Harry Smith, and Barbara A. Spicer pp 733 - 736; DOI: 10.1021/jm00241a018 |
|
Synthesis of an active hydroxylated glutethimide metabolite and some related analogs with sedative-hypnotic and anticonvulsant properties Hassan Y. Aboul-Enein, Charles W. Schauberger, Alfred R. Hansen, and Lawrence J. Fischer pp 736 - 741; DOI: 10.1021/jm00241a019 |
|
Synthesis and antihypertensive properties of new 3-hydrazinopyridazine derivatives Giorgio Pifferi, Francesco Parravicini, Carlo Carpi, and Luciano Dorigotti pp 741 - 746; DOI: 10.1021/jm00241a020 |
|
Quinoxaline studies. 23. Potential antimalarials. Substituted 5,8-dimethoxyquinoxalines George H. Fisher, Henry R. Moreno, John E. Oatis, and Harry P. Schultz pp 746 - 752; DOI: 10.1021/jm00241a021 |
|
Synthesis and antibacterial activities of some chloro analogs of 3-amino-3,4-dihydro-1-hydroxycarbostyril Alvie L. Davis, William H. Chambers, Don H. Kelley, David A. Fell, John R. Haynes, Karen L. Hulme, Larry D. Gage, and Tommy J. McCord pp 752 - 755; DOI: 10.1021/jm00241a022 |
|
Ellipticine derivatives Robert W. Guthrie, Arnold Brossi, Francis A. Mennona, John G. Mullin, Richard W. Kierstead, and E. Grunberg pp 755 - 760; DOI: 10.1021/jm00241a023 |
|
Bradykinin analogs containing .beta.-homoamino acids Miguel A. Ondetti and Stanford L. Engel pp 761 - 763; DOI: 10.1021/jm00241a024 |
|
Potential central nervous system antineoplastic agents. Amides of 6-cyano-6-norlysergic acid David E. Portlock, William C. Schwarzel, Anil C. Ghosh, Haldean C. Dalzell, and Raj K. Razdan pp 764 - 765; DOI: 10.1021/jm00241a025 |
|
Antifertility agents. 11. Secosteroids. 5. Synthesis of 9,11-secoestradiol Pannalal Kole, Suprabhat Ray, Ved P. Kamboj, and Nitya Anand pp 765 - 766; DOI: 10.1021/jm00241a026 |
|
Confirmation by synthesis of ristosamine as 3-amino-2,3,6-trideoxy-L-ribo-hexose William W. Lee, Helen Y. Wu, John J. Marsh, Carol W. Mosher, Edward M. Acton, Leon Goodman, and David W. Henry pp 767 - 768; DOI: 10.1021/jm00241a027 |
|
Confirmation by synthesis of the structure of acosamine and methyl N-acetylactinosaminide William W. Lee, Helen Y. Wu, J. E. Christensen, Leon Goodman, and David W. Henry pp 768 - 769; DOI: 10.1021/jm00241a028 |
|
Book Reviews pp 770 - 770; DOI: 10.1021/jm00241a600 |
|
Synthetic studies on nucleoside antibiotics. 13. Inhibitors of protein synthesis. 4. Structure-activity relation of gougerotin and some of its analogs C. Coutsogeorgopoulos, A. Bloch, K. A. Watanabe, and J. J. Fox pp 771 - 776; DOI: 10.1021/jm00242a001 |
|
Synthesis and biological activity of 10-thia-10-deaza analogs of folic acid, pteroic acid, and related compounds Y. H. Kim, Y. Gaumont, R. L. Kisliuk, and H. G. Mautner pp 776 - 780; DOI: 10.1021/jm00242a002 |
|
Synthesis and biological activities of some N6-(nitro- and -aminobenzyl)adenosines Shib P. Dutta, George L. Tritsch, Clifford Cox, and Girish B. Chheda pp 780 - 783; DOI: 10.1021/jm00242a003 |
|
Synthesis and biological activity of 5-fluoro-4'-thiouridine and some related nucleosides M. Bobek, A. Bloch, R. Parthasarathy, and R. L. Whistler pp 784 - 787; DOI: 10.1021/jm00242a004 |
|
Synthesis and pharmacology of 5-noralkyl-9.beta.-methyl-6,7-benzomorphans and stereochemistry of some intermediates Hirozumi Inoue, Tokuro Ohishi, and Everett L. May pp 787 - 791; DOI: 10.1021/jm00242a005 |
|
Microbial models of mammalian metabolism. O-Dealkylation of 10,11-dimethoxyaporphine J. P. Rosazza, A. W. Stocklinski, M. A. Gustafson, J. Adrian, and R. V. Smith pp 791 - 794; DOI: 10.1021/jm00242a006 |
|
Antiprotozoal thiazoles. 2-(5-Nitro-2-thienyl)thiazoles John P. Verge and Patrick Roffey pp 794 - 797; DOI: 10.1021/jm00242a007 |
|
Organic disulfides and related substances. 38. Disulfide and trisulfide sulfinate salts as antiradiation drugs Pramod K. Srivastava, Lamar Field, and Marie M. Grenan pp 798 - 802; DOI: 10.1021/jm00242a008 |
|
Hydroxy derivatives of S-2-(3-aminopropylamino)ethyl dihydrogen phosphorothioate and related compounds as antiradiation agents James R. Piper, Lucy M. Rose, Thomas P. Johnston, and Marie M. Grenan pp 803 - 812; DOI: 10.1021/jm00242a009 |
|
Antitumor agents. 16. Steroidal .alpha.-methylene-.gamma.-lactones Kuo-Hsiung Lee, Toshiro Ibuka, Sun-Hyuk Kim, Bruce R. Vestal, Iris H. Hall, and Eng-Shang Huang pp 812 - 817; DOI: 10.1021/jm00242a010 |
|
7.alpha.-Carboalkoxy steroidal spirolactones as aldosterone antagonists Richard M. Weier and Lorenz M. Hofmann pp 817 - 821; DOI: 10.1021/jm00242a011 |
|
Synthesis and some pharmacological properties of [3-.beta.-(2-thienyl)-L-alanine]-8-lysine-vasopressin Clark W. Smith, Martha F. Ferger, and W. Y. Chan pp 822 - 825; DOI: 10.1021/jm00242a012 |
|
Potential latentiation forms of biologically active compounds based on action of leucine aminopeptidase. Dipeptide derivatives of the tricycloaliphatic .alpha.-amino acid, adamantanine Herbert T. Nagasawa, James A. Elberling, and Frances N. Shirota pp 826 - 830; DOI: 10.1021/jm00242a013 |
|
Potential histamine H2-receptor antagonists. 2. N.alpha.-Guanylhistamine Graham J. Durant, Michael E. Parsons, and James W. Black pp 830 - 833; DOI: 10.1021/jm00242a014 |
|
Hypolipidemic imidazoles Keith H. Baggaley, Monique Heald, Richard M. Hindley, Brian Morgan, John L. Tee, and Joseph Green pp 833 - 836; DOI: 10.1021/jm00242a015 |
|
Conformational effects on the activity of drugs. 5. Pharmacological properties of 2-(p-nitrophenyl)-4-isopropylmorpholine, a cyclic analog of INPEA [1-(p-nitrophenyl)-2-isopropylaminoethanol] M. Del Tacca, A. Bertelli, L. Mazzanti, B. Stacchini, A. Balsamo, P. Crotti, B. Macchia, and F. Macchia pp 836 - 838; DOI: 10.1021/jm00242a016 |
|
Structure-activity relations in reactivators of organophosphorus-inhibited acetylcholinesterase. 9. N-Heterocyclic acraldoximes methiodides Palmarisa Franchetti, Mario Grifantini, and Sante Martelli pp 839 - 842; DOI: 10.1021/jm00242a017 |
|
Structure-activity relations in cinnamamides. 1. Synthesis and pharmacological evaluation of some (E)- and (Z)-N-alkyl-.alpha.,.beta.-dimethylcinnamamides A. Balsamo, P. L. Barili, P. Crotti, B. Macchia, F. Macchia, A. Pecchia, A. Cuttica, and N. Passerini pp 842 - 846; DOI: 10.1021/jm00242a018 |
|
Potential central nervous system antitumor agents. Hydantoin derivatives Geoffrey W. Peng, Victor E. Marquez, and John S. Driscoll pp 846 - 849; DOI: 10.1021/jm00242a019 |
|
Aromatic esters of 5-O-desosaminylerythronolide A oxime Ronald A. LeMahieu, Mathew Carson, Richard W. Kierstead, and Sidney Pestka pp 849 - 851; DOI: 10.1021/jm00242a020 |
|
Synthesis and antiarrhythmic activity of substituted (2-pyrimidinylthio)acetamidoximes Anthony C. Scotese, Arthur A. Santilli, and George L. Nelson pp 852 - 854; DOI: 10.1021/jm00242a021 |
|
Synthesis and analgesic activities of 2,5-dimethyl-2'-hydroxy-9.alpha.- and -.beta.-propyl-6,7-benzomorphans Kenner C. Rice, Arthur E. Jacobson, and Everette L. May pp 854 - 857; DOI: 10.1021/jm00242a022 |
|
Synthesis and neuroleptic activity of isomeric thieno[1,4]benzothiazines C. J. Grol and H. Rollema pp 857 - 861; DOI: 10.1021/jm00242a023 |
|
Book Reviews pp 861 - 864; DOI: 10.1021/jm00242a600 |
|
Calculation of hydrophobic constant (log P) from .pi. and f constants A. Leo, P. Y. C. Jow, C. Silipo, and C. Hansch pp 865 - 868; DOI: 10.1021/jm00243a001 |
|
Rm values of phenols. Their relation with log P values and activity G. L. Biagi, O. Gandolfi, M. C. Guerra, A. M. Barbaro, and G. Cantelli-Forti pp 868 - 873; DOI: 10.1021/jm00243a002 |
|
Rm values of steroids as an expression of their lipophilic character in structure-activity studies G. L. Biagi, A. M. Barbaro, O. Gandolfi, M. C. Guerra, and G. Cantelli-Forti pp 873 - 883; DOI: 10.1021/jm00243a003 |
|
Regression analysis of the relation between physical properties and the in vitro inhibition of monoamine oxidase by propynylamines Yvonne C. Martin, William B. Martin, and Julius D. Taylor pp 883 - 888; DOI: 10.1021/jm00243a004 |
|
Potential inhibitors of L-asparagine biosynthesis. 3. Aromatic sulfonyl fluoride analogs of L-asparagine and L-glutamine Michael Mokotoff, Steven Brynes, and James F. Bagaglio pp 888 - 891; DOI: 10.1021/jm00243a005 |
|
Ergot alkaloids. Synthesis of 6-methyl-8-ergolenes as inhibitors of prolactin release George S. Li, J. Michael Robinson, Heinz G. Floss, and John M. Cassady pp 892 - 895; DOI: 10.1021/jm00243a006 |
|
4-Trifluoromethylimidazoles and 5-(4-pyridyl)-1,2,4-triazoles, new classes of xanthine oxidase inhibitors J. J. Baldwin, P. A. Kasinger, F. C. Novello, J. M. Sprague, and D. E. Duggan pp 895 - 900; DOI: 10.1021/jm00243a007 |
|
3,5-Disubstituted 1,2,4-triazoles, a new class of xanthine oxidase inhibitor D. E. Duggan, R. M. Noll, J. E. Baer, F. C. Novello, and J. J. Baldwin pp 900 - 905; DOI: 10.1021/jm00243a008 |
|
Chemical differentiation of histamine H1- and H2-receptor agonists Graham J. Durant, C. Robin Ganellin, and Michael E. Parsons pp 905 - 909; DOI: 10.1021/jm00243a009 |
|
Methotrexate analogs. 6. Replacement of glutamic acid by various amino acid esters and amines Michael Chaykovsky, Barbara L. Brown, and E. J. Modest pp 909 - 912; DOI: 10.1021/jm00243a010 |
|
Potential filaricides. 6. Synthesis of 3,8-disubstituted 1,3,8-triazabicyclo[4.4.0]decan-2-ones and -thiones Satyavan Sharma, R. Bindra, R. N. Iyer, and Nitya Anand pp 913 - 917; DOI: 10.1021/jm00243a011 |
|
Potential bioreductive alkylating agents. 5. Antineoplastic activity of quinoline-5,8-diones, naphthazarins, and naphthoquinones Ai Jeng Lin, Brian J. Lillis, and Alan C. Sartorelli pp 917 - 921; DOI: 10.1021/jm00243a012 |
|
Antifertility agents. 8. Seco steroids. 2. 5,6-Secoestradiol and some related compounds Jasjit S. Bindra, A. T. Neyyarapally, R. C. Gupta, V. P. Kamboj, and Nitya Anand pp 921 - 925; DOI: 10.1021/jm00243a013 |
|
Oxanilic acids, a new series of orally active antiallergic agents John H. Sellstedt, Charles J. Guinosso, Albert J. Begany, Stanley C. Bell, and Marvin Rosenthale pp 926 - 933; DOI: 10.1021/jm00243a014 |
|
Synthesis of ethyl 6-substituted-chroman- and -chromone-2-carboxylates. Comparative structure-activity study employing the 6-phenyl and phenoxy analogs in the triton hyperlipidemic rat model Donald T. Witiak, William P. Heilman, Shankar K. Sankarappa, Richard C. Cavestri, and Howard A. I. Newman pp 934 - 942; DOI: 10.1021/jm00243a015 |
|
1-[[(5-Nitrofuranyl)methylene]amino]-4- and/or -5-substituted 2-imidazolidinones Harry R. Snyder, Leonard L. Bird, Arthur J. Siedler, and Jon Andersen pp 942 - 945; DOI: 10.1021/jm00243a016 |
|
Inhibitors of polyamine biosynthesis. 3. (+-)-5-Amino-2-hydrazino-2-methylpentanoic acid, an inhibitor of ornithine decarboxylase Mahmoud M. Abdel-Monem, Nancy E. Newton, and Charles E. Weeks pp 945 - 948; DOI: 10.1021/jm00243a017 |
|
Synthesis and biological properties of the 2-L-.beta.-(pyrazolyl-1)alanine analogs of luteinizing hormone-releasing hormone and thyrotropin-releasing hormone David H. Coy, Yoshihiro Hirotsu, Tommie W. Redding, Esther J. Coy, and Andrew V. Schally pp 948 - 949; DOI: 10.1021/jm00243a018 |
|
Structure-activity relation in synthetic fibrinolytics. 2-Phenethynylcyclopropanecarboxylates Masafumi Yoshimoto, Kurt N. Von Kaulla, and Corwin Hansch pp 950 - 951; DOI: 10.1021/jm00243a019 |
|
Benzoxocin and benzoxonin derivatives. Novel groups of terpenophenols with central nervous system activity. Correction Shlomo Houry, Raphael Mechoulam, and Bernard Loev pp 951 - 952; DOI: 10.1021/jm00243a020 |
|
Synthesis and hypoglycemic activity of phenacyltriphenylphosphoranes and phosphonium salts Benjamin Blank, Nicholas W. DiTullio, Linda Deviney, John T. Roberts, and Harry L. Saunders pp 952 - 954; DOI: 10.1021/jm00243a021 |
|
Preparation and biological activity of some aminoacyl and peptidyl derivatives of 2'-amino-2'-deoxyuridine R. A. Sharma, M. Bobek, and A. Bloch pp 955 - 957; DOI: 10.1021/jm00243a022 |
|
Book Reviews pp 957 - 958; DOI: 10.1021/jm00243a600 |
|
Noncomputer approach to structure-activity study. Expanded Fibonacci search applied to structurally diverse types of compounds Norman J. Santora and King Auyang pp 959 - 963; DOI: 10.1021/jm00244a001 |
|
Role of anionic, imidic, and amidic forms in structure-activity relations. Correlation of electronic indexes and bacteriostatic activity in sulfonamides Augusto Rastelli, Pier G. De Benedetti, Giovanna Gavioli Battistuzzi, and Albano Albasini pp 963 - 967; DOI: 10.1021/jm00244a002 |
|
Inhibitors of nucleoside transport. Structure-activity study using human erythrocytes Brajeswar Paul, Marianne F. Chen, and Alan R. P. Paterson pp 968 - 973; DOI: 10.1021/jm00244a003 |
|
Synthesis and cell culture studies on the antiviral activity of 5-mercaptomethyl-2'-deoxyuridine V. S. Gupta, G. L. Bubbar, J. B. Meldrum, and J. R. Saunders pp 973 - 976; DOI: 10.1021/jm00244a004 |
|
Synthesis and central nervous system effects of 8,9-dihydro[1]benzazepino[3,2,1-jk][1,4]benzodiazepin-1(2H)-ones and [1]benzazepino[3,2,1-jk][1,4]benzodiazepin-1(2H)-ones Luciano Toscano, Ennio Seghetti, and Giuseppe Fioriello pp 976 - 981; DOI: 10.1021/jm00244a005 |
|
Flavonoids. 8. Synthesis and antifertility and estrogen receptor binding activities of coumarins and .DELTA.3-isoflavenes Mansukh C. Wani, Douglas H. Rector, H. Dix Christensen, Gary L. Kimmel, and Clarence E. Cook pp 982 - 985; DOI: 10.1021/jm00244a006 |
|
Chemistry of cephalosporin antibiotics. 28. Preparation and biological activity of 3-(substituted)vinyl cephalosporins J. Alan Webber, John L. Ott, and Robert T. Vasileff pp 986 - 992; DOI: 10.1021/jm00244a007 |
|
9-Chloro-2,3-dihydro-5H-1,4-dioxepino[6,5-b]benzofuran, a novel antilipidemic agent structurally related to clofibrate Donald T. Witiak, Guiragos K. Poochikian, Dennis R. Feller, Nancy A. Kenfield, and Howard A. I. Newman pp 992 - 996; DOI: 10.1021/jm00244a008 |
|
Stereoisomeric 5,9-dimethyl-2'-hydroxy-2-tetrahydrofurfuryl-6,7-benzomorphans, strong analgesics with nonmorphinelike action profiles Herbert Merz, Klaus Stockhaus, and Helmut Wick pp 996 - 1000; DOI: 10.1021/jm00244a009 |
|
Emetic activity of N-substituted norapomorphines Edward R. Atkinson, Francis J. Bullock, Felix E. Granchelli, Sydney Archer, Franklin J. Rosenberg, David G. Teiger, and Frederick C. Nachod pp 1000 - 1003; DOI: 10.1021/jm00244a010 |
|
Alkylating derivatives of amino acids and peptides. Synthesis of N-maleoylamino acids, [1-(N-maleoylglycyl)cysteinyl]oxytocin, and [1-(N-maleoyl-11-aminoundecanoyl)cysteinyl]oxytocin. Effects on vasopressin-stimulated water loss from isolated toad bladder Daniel H. Rich, Paul D. Gesellchen, Alex Tong, Al Cheung, and Carl K. Buckner pp 1004 - 1010; DOI: 10.1021/jm00244a011 |
|
Antimalarial phenanthrene amino alcohols. 3. Halogen-containing 9-phenanthrenemethanols Edward A. Nodiff, Andrew J. Saggiomo, Keiichi Tanabe, Eugene H. Chen, Masafu Shinbo, Mahesh P. Tyagi, Atsuto Kozuka, Hirotaka Otomasu, Basant L. Verma, and David Goff pp 1011 - 1019; DOI: 10.1021/jm00244a012 |
|
Synthesis and pharmacological properties of [1-L-penicillamine,4-L-leucine]oxytocin Martha F. Ferger and W. Y. Chan pp 1020 - 1022; DOI: 10.1021/jm00244a013 |
|
[4-Phenylalanine]oxytocin, an inhibitor of the antidiuretic effect of 8-arginine-vasopressin John J. Nestor, Martha F. Ferger, and W. Y. Chan pp 1022 - 1024; DOI: 10.1021/jm00244a014 |
|
Cycloalkanones. 7. Hypocholesterolemic activity of aliphatic compounds related to 2,8-dibenzylcyclooctanone G. L. Carlson, I. H. Hall, and C. Piantadosi pp 1024 - 1026; DOI: 10.1021/jm00244a015 |
|
trans-2-Acetoxycyclobutyltrimethylammonium iodide, a cyclobutane analog of trans-ACTM [trans-2-acetoxycyclopropyltrimethylammonium iodide] Joseph G. Cannon, Theresa Lee, V. Sankaran, and John Paul Long pp 1027 - 1028; DOI: 10.1021/jm00244a016 |
|
Preparation of nitroso-13N-labeled nitrosoureas William A. Pettit, Richard H. Mortara, George A. Digenis, and Mary F. Reed pp 1029 - 1031; DOI: 10.1021/jm00244a017 |
|
3-Hydroxymethyl-s-triazolo[3,4-a]phthalazine, a novel urinary hydralazine metabolite in man Hans Zimmer, Robert Glaser, John Kokosa, Daniel A. Garteiz, Evelyn V. Hess, and A. Litwin pp 1031 - 1033; DOI: 10.1021/jm00244a018 |
|
Preparation and analgesic activity of 3,6-diacetylnormorphine and 6-acetylnormorphine Kenner C. Rice and Arthur E. Jacobson pp 1033 - 1035; DOI: 10.1021/jm00244a019 |
|
Analgetic activity and in vitro binding constants of some N-alkyl-3-benzazocines Michael E. Rogers, Helen H. Ong, Everette L. May, and Werner A. Klee pp 1036 - 1038; DOI: 10.1021/jm00244a020 |
|
Synthesis and antibacterial evaluation of 1,2,3,4-tetrahydro-4-oxo-1,8-naphthyridine-3-carboxylic acid esters, carbonitriles, and carboxamides Arthur A. Santilli, Anthony C. Scotese, and John A. Yurchenco pp 1038 - 1041; DOI: 10.1021/jm00244a021 |
|
Synthesis of tritium- and deuterium-labeled 9-.beta.-D-arabinofuranosyladenine and the tritium-labeled 5'-monophosphate ester with increased metabolic stability David C. Baker and Theodore H. Haskell pp 1041 - 1044; DOI: 10.1021/jm00244a022 |
|
[1-.beta.-Mercaptopropionic acid,2-(3,5-dibromo-L-tyrosine)]oxytocin, a potent inhibitor of oxytocin Edwin O. Lundell and Martha F. Ferger pp 1045 - 1047; DOI: 10.1021/jm00244a023 |
|
Book Reviews pp 1047 - 1050; DOI: 10.1021/jm00244a600 |
|
Quantum chemical studies of meperidine and prodine Gilda H. Loew and J. Randal Jester pp 1051 - 1056; DOI: 10.1021/jm00245a001 |
|
Hydrophobic binding site in acetylcholinesterase George M. Steinberg, Morton L. Mednick, Jan Maddox, Robert Rice, and Joyce Cramer pp 1056 - 1061; DOI: 10.1021/jm00245a002 |
|
Primary and .beta.-secondary deuterium isotope effects in N-deethylation reactions Sidney D. Nelson, Lance R. Pohl, and William F. Trager pp 1062 - 1065; DOI: 10.1021/jm00245a003 |
|
Hypo-.beta.-lipoproteinemic agents. 1. Bicyclo[2.2.2]octyloxyaniline and its derivatives Charles E. Day, Paul E. Schurr, D. Edward Emmert, Ruth E. TenBrink, and Daniel Lednicer pp 1065 - 1070; DOI: 10.1021/jm00245a004 |
|
Nucleic acid related compounds. 17. 3-Deazauridine. Stannous chloride catalysis of cis-diol vs. phenolic base methylation with diazomethane Morris J. Robins and Alan S. K. Lee pp 1070 - 1074; DOI: 10.1021/jm00245a005 |
|
Synthesis of thebaine and oripavine from codeine and morphine Randy B. Barber and Henry Rapoport pp 1074 - 1077; DOI: 10.1021/jm00245a006 |
|
Cardiovascular activity of aromatic guanidine compounds John L. Hughes, R. C. Liu, T. Enkoji, Carroll M. Smith, James W. Bastian, and Pedro D. Luna pp 1077 - 1088; DOI: 10.1021/jm00245a007 |
|
Synthesis of a bifunctional coordination complex of osmium with curariform activity Dermot B. Taylor, Kenneth P. Callahan, and Iqbal Shaikh pp 1088 - 1094; DOI: 10.1021/jm00245a008 |
|
Synthesis and biological properties of some novel heterocyclic homoprostanoids A. Douglas Bender, Charles E. Berkoff, William G. Groves, Linda M. Sofranko, George R. Wellman, Jih-Hua Liu, Peter P. Begosh, and Joseph W. Horodniak pp 1094 - 1098; DOI: 10.1021/jm00245a009 |
|
Synthesis and antitumor activity of 2-deamino- and N2-(.gamma.-hydroxypropyl)actinomycin D Stanley Moore, Michio Kondo, Michelle Copeland, Johannes Meienhofer, and Randall K. Johnson pp 1098 - 1101; DOI: 10.1021/jm00245a010 |
|
Synthesis of deuterium-labeled analogs of cyclophosphamide and its metabolites Leslie J. Griggs and Michael Jarman pp 1102 - 1106; DOI: 10.1021/jm00245a011 |
|
Synthesis and antitumor activity of 6-trifluoromethylcyclophosphamide and related compounds Peter B. Farmer and Peter J. Cox pp 1106 - 1110; DOI: 10.1021/jm00245a012 |
|
Potential antitumor agents. 16. 4'-(Acridin-9-ylamino)methanesulfonanilides Bruce F. Cain, Graham J. Atwell, and William A. Denny pp 1110 - 1117; DOI: 10.1021/jm00245a013 |
|
Antiallergic activity of 2-phenyl-8-azapurin-6-ones B. J. Broughton, P. Chaplen, P. Knowles, E. Lunt, S. M. Marshall, D. L. Pain, and K. R. H. Wooldridge pp 1117 - 1122; DOI: 10.1021/jm00245a014 |
|
Antimalarials. 7. 2,8-Bis(trifluoromethyl)-4-quinolinemethanols Peter Blumbergs, Meng-Sheng Ao, Maurice P. LaMontagne, Anica Markovac, Jaroslav Novotny, Carol H. Collins, and Fred W. Starks pp 1122 - 1126; DOI: 10.1021/jm00245a015 |
|
3-Arylquinolizidines, potential antidepressant agents M. E. Rogers and Joseph Sam pp 1126 - 1130; DOI: 10.1021/jm00245a016 |
|
Antiarrhythmics. N-(Aminoalkylene)trifluoroethoxybenzamides and N-(aminoalkylene)trifluoroethoxynaphthamides E. H. Banitt, W. E. Coyne, J. R. Schmid, and A. Mendel pp 1130 - 1134; DOI: 10.1021/jm00245a017 |
|
Alkylating analogs of bradykinin John Turk, Philip Needleman, and Garland R. Marshall pp 1135 - 1139; DOI: 10.1021/jm00245a018 |
|
Analogs of bradykinin with restricted conformational freedom John Turk, Philip Needleman, and Garland R. Marshall pp 1139 - 1142; DOI: 10.1021/jm00245a019 |
|
17.alpha.-Ethyl-20.alpha.- and -20.beta.-dihydroprogesterones and other 17.alpha.-ethyl-substituted pregnanes as potential contragestational agents Ramesh M. Kanojia, Paul Ostrowski, Do Won Hahn, George Allen, and John L. McGuire pp 1143 - 1145; DOI: 10.1021/jm00245a020 |
|
2-(3,4-Dichloroanilino)quinolizinium bromide, a unique antispasmodic, antisecretory, and antiulcerogenic agent Robert J. Alaimo and Marvin M. Goldenberg pp 1145 - 1147; DOI: 10.1021/jm00245a021 |
|
Structure-activity relations in reactivators of organophosphorus-inhibited acetylcholinesterase. 10. Hydroxyiminomethylarylethenylpyridine methiodides Francesca Arena, Fedele Manna, Cosimo Pizza, Maria Luisa Stein, and Mario Grifantini pp 1147 - 1150; DOI: 10.1021/jm00245a022 |
|
Platinum complex inhibition of leucine aminopeptidase Paul Melius and C. A. McAuliffe pp 1150 - 1151; DOI: 10.1021/jm00245a023 |
|
Application of the carbonic anhydrase inhibitory effect of furosemide to the study of furosemide release from two of its diuretic derivatives Gil Navon, Jashovam Shani, Ruth Panigel, and Shlomo Schoenberg pp 1152 - 1154; DOI: 10.1021/jm00245a024 |
|
Growth inhibitory properties of aromatic .alpha.-ketoaldehydes toward bacteria and yeast. Comparison of inhibition and glyoxalase I activity David L. Vander Jagt pp 1155 - 1158; DOI: 10.1021/jm00245a025 |
|
Synthesis and antiinflammatory activity of some 2-heteroaryl-.alpha.-methyl-5-benzoxazoleacetic acids David W. Dunwell, Delme Evans, and Terence A. Hicks pp 1158 - 1159; DOI: 10.1021/jm00245a026 |
|
Lapachol derivative active against mouse lymphocytic leukemia P-388 M. da Consolacao F. Linardi, M. M. De Oliveira, and M. R. P. Sampaio pp 1159 - 1161; DOI: 10.1021/jm00245a027 |
|
Nonclassical nicotine antagonists Charles F. Barfknecht, Clinton A. Taylor, Lawrence A. Peterson, Fouad M. Sharabi, and John P. Long pp 1161 - 1164; DOI: 10.1021/jm00245a028 |
|
Methyl 5(6)-phenylsulfinyl-2-benzimidazolecarbamate, a new, potent anthelmintic Eugene A. Averkin, Colin C. Beard, Charles A. Dvorak, John A. Edwards, John H. Fried, John G. Kilian, Richard A. Schiltz, Theodore P. Kistner, J. H. Drudge, and et al. pp 1164 - 1166; DOI: 10.1021/jm00245a029 |
|
Synthesis and antibacterial properties of methylsulfinyl and methylsulfonyl analogs of some nitrofurans Bertil Ekstrom, Maria Ovesson, and Brian G. Pring pp 1166 - 1168; DOI: 10.1021/jm00245a030 |
|
Book Reviews pp 1168 - 1174; DOI: 10.1021/jm00245a600 |
|
7-Substituted actinomycin D analogs. Chemical and growth-inhibitory studies S. K. Sengupta, S. K. Tinter, H. Lazarus, B. L. Brown, and E. J. Modest pp 1175 - 1180; DOI: 10.1021/jm00246a001 |
|
Synthesis and evaluation of [des-Asp1]angiotensin I as a precursor for [des-Asp1]angiotensin II (angiotensin III) B. S. Tsai, M. J. Peach, M. C. Khosla, and F. M. Bumpus pp 1180 - 1183; DOI: 10.1021/jm00246a002 |
|
Synthesis of lysophosphatidylethanolamine analogs that inhibit renin activity Joseph G. Turcotte, Cheng-Sein Yu, Hwei-Ling Lee, Sripada K. Pavanaram, Subha Sen, and Robert R. Smeby pp 1184 - 1190; DOI: 10.1021/jm00246a003 |
|
Quinazolines as inhibitors of dihydrofolate reductase. 3. Analogs of pteroic and isopteroic acids John B. Hynes, John M. Buck, Leo D'Souza, and James H. Freisheim pp 1191 - 1194; DOI: 10.1021/jm00246a004 |
|
Cholinergic effects of molecular segments of apomorphine and dopaminergic effects of N,N-dialkylated dopamines James Z. Ginos, Geurge C. Cotzias, Eduardo Tolosa, Lily C. Tang, and Anthony LoMonte pp 1194 - 1200; DOI: 10.1021/jm00246a005 |
|
Psychotomimetic phenylisopropylamines. 5. 4-Alkyl-2,5-dimethoxyphenylisopropylamines Alexander T. Shulgin and Donald C. Dyer pp 1201 - 1204; DOI: 10.1021/jm00246a006 |
|
Novel phosphate anthelmintics. 3. Alkyl and aryl 1-methyleneallyl phosphates, phosphonates, and phosphinates Kurt Pilgram and D. Kendall Hass pp 1204 - 1211; DOI: 10.1021/jm00246a007 |
|
N-Isopropyl derivatives of dopamine and 5,6-dihydroxy-2-aminotetralin Joseph G. Cannon, John P. O'Donnell, Theresa Lee, Charles R. Hoppin, John Paul Long, Mustafa Ilhan, Brenda Costall, and Robert J. Naylor pp 1212 - 1216; DOI: 10.1021/jm00246a008 |
|
Antimalarials. Synthesis and antimalarial activity of 1-(4-methoxycinnamoyl)-4-(5-phenyl-4-oxo-2-oxazolin-2-yl)piperazine and derivatives Thomas R. Herrin, Jeanne M. Pauvlik, Evelyn V. Schuber, and Adolph O. Geiszler pp 1216 - 1223; DOI: 10.1021/jm00246a009 |
|
Antimalarials. 3. 3-Substituted 1-naphthalenemethanols J. Samuel Gillespie, Satya P. Acharya, Dwight A. Shamblee, and Richard E. Davis pp 1223 - 1227; DOI: 10.1021/jm00246a010 |
|
Structure-activity relations of antiarrhythmic 6-substituted decahydroisoquinolines Ian W. Mathison and Richard R. Tidwell pp 1227 - 1231; DOI: 10.1021/jm00246a011 |
|
Antimalarials. 10. Substituted 3-halo- and 3-methoxy-2-aryl-4-quinoline(dibutylaminomethyl)methanols H. Randall Munson, Richard E. Johnson, J. Milton Sanders, Cyrus J. Ohnmacht, and Robert E. Lutz pp 1232 - 1236; DOI: 10.1021/jm00246a012 |
|
Synthesis of 5-amino-1-(5-deoxy-.beta.-D-ribofuranosyl)imidazole-4-carboxamide and related 5'-deoxyimidazole ribonucleosides Prem C. Srivastava, Arthur R. Newman, Thomas R. Matthews, and Roland K. Robins pp 1237 - 1240; DOI: 10.1021/jm00246a013 |
|
1-Substituted 4-(1,2-diphenylethyl)piperazine derivatives and their analgesic activities. 1 Kagayaki Natsuka, Hideo Nakamura, Hitoshi Uno, and Susumu Umemoto pp 1240 - 1244; DOI: 10.1021/jm00246a014 |
|
Antagonism of luteinizing hormone release and of ovulation by an analog of the luteinizing hormone-releasing hormone John P. Yardley, Theodore J. Foell, Craig Beattie, and Norman H. Grant pp 1244 - 1247; DOI: 10.1021/jm00246a015 |
|
Luteinizing hormone-releasing hormone. Antiovulatory activity of analogs substituted in positions 2 and 6 C. W. Beattie, A. Corbin, T. J. Foell, V. Garsky, W. A. McKinley, R. W. A. Rees, D. Sarantakis, and J. P. Yardley pp 1247 - 1250; DOI: 10.1021/jm00246a016 |
|
Synthesis and antitumor activity of cyclophosphamide analogs. 1. Benzo annulated cyclophosphamide and related systems Susan M. Ludeman and Gerald Zon pp 1251 - 1253; DOI: 10.1021/jm00246a017 |
|
Synthesis and antimicrobial activity of certain imidazo[1,2-a]pyrimidines Ganapathi R. Revankar, Thomas R. Matthews, and Roland K. Robins pp 1253 - 1255; DOI: 10.1021/jm00246a018 |
|
Synthesis of some glycoside analogs and related compounds from 9-amino-6-(methylthio)-9H-purine Carroll Temple, Conrad L. Kussner, and John A. Montgomery pp 1255 - 1258; DOI: 10.1021/jm00246a019 |
|
Synthesis of 6.alpha.-methyldigitoxigenin 3-acetate Umberto Valcavi, Bruno Corsi, Roberto Caponi, Sergio Innocenti, and Paola Martelli pp 1258 - 1261; DOI: 10.1021/jm00246a020 |
|
Synthesis and some pharmacological properties of [1-.beta.-mercapto-.beta.,.beta.-diethylpropionic acid,2-(3,5-dibromo-L-tyrosine)]oxytocin Edwin O. Lundell, Clark W. Smith, and Martha F. Ferger pp 1262 - 1264; DOI: 10.1021/jm00246a021 |
|
3-Acyloxymethyl-7-(2-thienylacetamido)-3-cephem-4-carboxylic acids. Improved synthesis and biological properties David A. Berges pp 1264 - 1265; DOI: 10.1021/jm00246a022 |
|
2,3,4,5,6,7-Hexahydro-1,6-methano-1H-3-benzazonine derivatives as analgesics Shunsaku Shiotani, Tadashi Kometani, and Kemmotsu Mitsuhashi pp 1266 - 1267; DOI: 10.1021/jm00246a023 |
|
Absolute configuration of the major metabolite of 5,5-diphenylhydantoin,5-(4'-hydroxyphenyl)-5-phenylhydantoin Jacques H. Poupaert, Robert Cavalier, Michel H. Claesen, and Pierre A. Dumont pp 1268 - 1271; DOI: 10.1021/jm00246a024 |
|
Molecular connectivity. 4. Relations to biological activities Lemont B. Kier, Wallace J. Murray, and Lowell H. Hall pp 1272 - 1274; DOI: 10.1021/jm00246a025 |
|
Additions and Corrections - Quinuclidine Chemistry. 3. β-cis-2-(4'-Chlorobenzhydryl)-3-quinuclidinol, a New Central Nervous System Stimulant. Importance of he Benzhydryl Configuration. E. J. Warawa, N. J. Mueller, and Jonas A. Gylys pp 1275 - 1275; DOI: 10.1021/jm00246a600 |
|
Additions and Corrections - Linear Regression Analysis of Inhibitroy Potency of Organic Disulfides against Histoplasma capsulatum L. J .Schaad, R. H .Werner, Lynn Dillon, Lamar Field, and C. Emory Tate pp 1275 - 1275; DOI: 10.1021/jm00246a601 |
|
Additions and Corrections - Synthesis of a Fluorescent Derivative of Amethopterin. G. R .Gapski, J. M .Whitely, J. I .Rader, P. L .Cramer, G. B. Henderson, V. Neef, and F. M. Huennekens pp 1275 - 1275; DOI: 10.1021/jm00246a602 |
|
Additions and Corrections - Studies in Antifertility Agents. 11. Secosteroids. 5. Synthesis of 9,11-Secoestradiol. Pannalal Kole, Suprabhat Ray, Ved P. Kamboj, and Nitya Anand pp 1275 - 1275; DOI: 10.1021/jm00246a603 |
|
Book Reviews pp 1275 - 1279; DOI: 10.1021/jm00246a604 |